Dose/day | Cmax (ng/ml) | Cmin (ng/ml) | |
Bosutinib | Probably does not require monitoring | ||
Dasatinib | 100 mg/day (QD) | >50 (efficacy) | <2.5 (tolerance) |
Imatinib | 400 mg/day (QD) | >1000 (efficacy) >3000 (tolerance) | |
Nilotinib | 600 mg/day (BID) | 800 (efficacy) | |
Ponatinib | No information |